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Pain-Relieving Rubs

All you knead

Oh, my aching fill-in-the-blank! There are so many different ways to hurt, and just as many ways to seek relief. But when RICE (Rest, Ice, Compression, and Elevation) just isn't doing the trick, you can try something stronger -- external counterirritants.

By stimulating receptors in the skin, counterirritants create a sensation of cold and/or warmth in the affected area, increasing blood flow and helping relieve discomfort. So lay your hands on a sore spot and work in the stuff. You'll feel better soon.


Managing Those Pesky Aches

Pain is pain, but pain relievers act differently. It appears that aspirin and other salicylates applied to the skin don't have much effect in relieving pain. Your primary methods of action against external pain are local analgesics, anesthetics, and counterirritants.

  • Counterirritants can be used with non-steroidal anti-inflammatory drugs (NSAIDs) or aspirin.
Analgesics and anesthetics block pain sensation by acting directly on the pain sensors in the skin. Counterirritants create sensations of warmth or cold, overloading sensors so they temporarily block out pain.

  • Topical liniments in an alcohol base penetrate more deeply into the skin than other vehicles. However, they can be more irritating to the skin.
  • Gels usually deliver a sense of warmth and penetrate the skin faster than lotions. They can cause a slight burning sensation, so do not exceed recommended dosage.
  • Heat increases the absorption of these liniments; be very careful in administering these topical drugs on a hot day or with the use of a heating pad.
  • Bandaging injuries tightly after applying counterirritants can cause irritation and blistering because the ingredients remain in contact with the skin for a longer period of time.
  • Capsaicin, a slow-acting counterirritant, is often combined with other agents to provide both slow and long-lasting relief. Capsaicin's pain-relieving effects can take from two to six weeks to occur.
  • The act of massaging agents on an injury often offers some temporary pain relief. Be aware, though, that rubbing them too vigorously into the skin can cause increased action of the ingredients and a burning sensation.

Topical anesthetics

Temporarily relieve pain, burning, itching, and discomfort by suppressing transmission of nerve impulses. Careful: these drugs may be absorbed into the bloodstream and cause toxic reactions when applied to broken skin. Take care to use these products sparingly and externally only.

Counterirritants

Reduce the perception of pain by stimulating the sensory nerve endings in the skin to produce the sensation of cooling or warming. The theory is that by producing this smaller irritation, you will be distracted from the greater pain.


Topical Anesthetics
Ingredient
Description
Benzocaine Very safe and effective in treating pain and itch. Has fewer side effects than the other "-caine" anesthetics because it is absorbed less easily. Provides relief for four to six hours.
Benzyl Alcohol Safe and effective in relieving itching and burning due to cuts and insect bites. Faster acting and shorter lasting than benzocaine.
Dibucaine Fast acting; effects last up to four hours. Very potent; do not use on broken skin or large areas.
Lidocaine Fast acting; effects last for several hours. Very potent; do not use on broken skin or large areas.
Pramoxine Safe and effective when used on unbroken skin.
Counterirritants
Ingredient
Description
Allyl Isothiocyanate (mustard plaster) A powerful irritant, but safe and effective. Blistering may occur in some cases. Do not use more than four times a day.
Ammonia Safe and effective. Blistering may occur in some cases. Do not use more than four times a day.
Camphor At concentrations of 0.1% to 3.0%, used as a topical pain reliever and anesthetic. In concentrations over 3%, induces relief of pain and discomfort by stimulating nerve endings. High doses are not recommended, as camphor is toxic.
Capsicum Preparations Creates a warm feeling but does not redden skin. Requires repeated use for maximum benefit. Safe and effective. Do not use more than four times a day.
Histamine Safe and effective when applied topically. Do not use more than three or four times daily.
Menthol Usually combined with other ingredients with analgesic properties, like camphor. Menthol causes sensitization in some people, although the sensitization index is low. Symptoms include urticaria, erythemia, and other cutaneous lesions, like contact dermititis.
Methyl Nicotinate Derived from the vitamin niacin. Safe and effective.
Methyl Salicylate Widely used in counterirritants. Very effective and safe. Poisonous if taken orally.
Turpentine Oil Turpentine is a potent skin irritant. Some people may experience allergic reactions. It has, however, been approved as safe and effective.

FDA-Approved Uses

Counterirritants
  • For the temporary relief of minor aches and pains of muscles and joints associated with simple backaches, arthritis, strains, bruises, and sprains.
Managing Minor Pain
  • Counterirritants should only be used over intact, unbroken skin to prevent systemic absorption.
  • Counterirritants can be used over the affected area up to four times per day.
  • Simply rub a thin layer of solution over the affected area.
RICE: the First Line for Injury
  • If you're treating an injury: Rest, Ice, Compress, Elevation.
  • Rest: do not use or move the injured area.
  • Ice: use in the first 24 hours after injury to reduce swelling.
  • Compress: wrapping the area in bandages further reduces swelling.
  • Elevation: raise the joint to reduce swelling.
See Your Doctor
  • For serious sprains and strains, consult your physician.

Warnings

Counterirritants

Consult a physician before using or do not use if you have:
  • Allergy to any counterirritants or aspirin
  • Skin conditions such as psoriasis or eczema
Or if you:
  • Are pregnant or are a nursing mother
  • Are administering to a child or infant
  • Plan to apply to wounds, lesions, broken, damaged, or sensitive skin
  • Plan to apply near eyes or other mucous membranes
Common Side Effects

Counterirritants
  • None anticipated
Infrequent to Rare Side Effects

  • Allergic skin rash
  • Skin irritation
Effects of Overdose

  • Overdose from topical use is not anticipated. Do not swallow.
What to Do in Case of Overdose

  • For external use only. If swallowed, immediately seek medical attention.

Websites, Organizations & Manufacturers
Sources & Further Reading

Government Sources

1. Food & Drug Administration.Federal Register 2/8/83.
2. Food & Drug Administration.Federal Register 7/30/86.
3. Food & Drug Administration.Federal Register 8/25/88.
Books

1. Covington, TR et al. Handbook of Nonprescription Drugs, Eleventh Ed. American Pharmaceutical Assoc. Washington, DC 1996.
2. Kastrup EK et al. Drug Facts and Comparisons. Facts and Comparisons.
3. Inlander, CB and Slamans, S.The Over-the-Counter Doctor. Cader Books. New York, NY 1997.
4. Zimmerman, DR.Zimmerman's Complete Guide to Nonprescription Drugs, Second Ed. Gale Research, Inc. 1983.
Find more books on health and wellness at barnesandnoble.com.

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